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Celecoxib (SC 58635) | 购买COX 抑制剂 - Selleck
来自 : 发布时间:2024-05-09
定制您的化合物库 通过在我们的库存中挑选化合物来建立合适的化合物库,用于您的研究工作。 您可以选择: 特定化合物 96/384孔板位图 可选择\"干/固体”或\"DMSO溶液” 请通过info@selleck.cn与我们联系,定制你所需要的化合物库。 今日订购,明日送达,全国免运费!全国免费电话:400-668-6834|Email:info@selleck.cn 在体外, Celecoxib有效选择性抑制COX-2,IC50为40 nM, 而作用于COX-1时,IC50为15 μM。[1]Celecoxib 作用于鼻咽癌 (NPC)细胞系,包括 HNE1和CNE1-LMP1,具有抗增殖效果,IC50分别为32.86 μM 和 61.31 μM。[4] M4H4U4lvHWlZYOgTWNCVS1zIHX4dJJme3Orb36gc44h[m:2aDDwdo91WmwIHHu[EBuWk6DIHzleoVt MoizQIEhfGG{Z3X0QUdg[myjbnunJIhzWZ;J3j0eJB{Qi9xcIXicYVlNm6lYnmucoxuNm6raD7nc5YwOjZ3MUOxO|IoRjJ4NUGzNVczRC:jPh?= MYpcoR2[2W|IFnDRW0uOSCneIDy[ZN{cW:wIH;uJIJwfGhicILveIVqdiCjbnSgcXJPSSCuZYlcC= NXzMR21oRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:vdJVjdWWmLn7jZokvdmyvLn7pbE5od3ZxMk[1NVMyPzJpPkK2OVE{OTd{PD;hQi= MYDzbYdvcW[rY3HueIx6KGmwY4LlZZNmeyC2aHWgTWM2OMLidnHseYV{KG:oIH;4ZYxqeGyjdHnuxsA NUHDdIZsRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:vdJVjdWWmLn7jZokvdmyvLn7pbE5od3ZxMk[0O|Q3QTNpPkK2OFc1Pjl|PD;hQi= NVnpOmVYe2mpbnnmbYNidnSueTDpcoNzWG|ZYOgeIhmKEmFNUFCpJZidHWnczDv[kBwgGGuaYDsZZRqdsLi M2j0d|xiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4D1Zo1mC6wY3LpMo5tdS6waXiu[493NzJ4NEe0Olk{Lz5{NkS3OFY6OzxxYU6= NWGWIdoemWmdXPld{BwgGGuaYDsZZRqdi2rbnT1Z4VlKGGyb4D0c5Nqew ? 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Celecoxib decreased protein expression of COX-2 compared with control as indicated by western blot. 在体内, Celecoxib 具有有效的口服抗炎活性。Celecoxib 降低卡拉胶水肿检测中的急性炎症,也降低佐剂性关节炎模型中的慢性炎症,ED50分别为7.1 mg/kg和 0.37 mg/kg/day。此外, Celecoxib作用于Hargreaves 痛模型,也具有镇痛活性,ED50为34.5 mg/kg。此外, Celecoxib 按200 mg/kg剂量处理大鼠,不会产生急性GI毒性,每天按600 mg/kg剂量处理大鼠,持续10天以上,不会产生GI毒性。[1]13.5 Gy 局部胸部照射(LTI)142天(范围为 94-155 天)后,Celecoxib 作用于C3Hf/KamLaw 雌性小鼠模型,提高105天的平均寿命 (范围为79-145 天)。[5] 体外COX酶实验 : 细胞匀浆与COX-1或COX-2杆状病毒温育3天,通过测评PG合成能力,而测定昆虫细胞中COX蛋白表达。搅匀表达COX-1或COX-2的细胞,然后与花生四烯酸 (10 μM)混合。通过监测PG产量,而测定COX活性。在模拟感染的Sf9细胞中检测不出COX活性。Celecoxib与天然1% CHAPS 匀浆(2-10 μg 蛋白)预温育10分钟,然后加入花生四烯酸。温育10分钟后,通过ELISA检测形成的PGE2。 Incubation Time: 48 小时 Method: 使用MTT实验测定 Celecoxib 作用于 NPC细胞的抗增殖效果。细胞接种在96孔板上,粘附24小时。使用浓度不断增高的Celecoxib (0 到 75 μM) (溶于 DMSO, 终浓度 ≤0.1%)处理细胞,然后再温育48小时。 温育后,每孔加入 20 μL MTT 染料 (5 mg/mL) ,然后在37oC下温育4小时。移除上清液,晶体溶解在 DMSO 中,然后在490 nm处测定吸光值。使用 Probit回归模型及SPSS 15.0 软件计算IC50值和95%置信区间。每组实验至少重复进行三次。(Only for Reference) Animal Models: 溶于0.9%生理盐水的0.1 mL 1%卡拉胶溶液或溶于50 μL 矿物油的1 mg 乳酸分枝杆菌注射到雄性Sprague−Dawley大鼠右后腿足垫 Dosages: ≤200 mg/kg Administration: 口服处理(Only for Reference) 从左到右依次将纯溶剂加入产品,现配现用(数据来自Selleck实验检测而非文献): 2% DMSO+30% PEG 300+5% Tween 80+ddH2O * 溶解度检测是由Selleck技术部门检测的,可能会和文献中提供的溶解度有所差异,这是由于生产工艺和批次不同产生的正常现象。请按照顺序依次加入各个纯溶剂。 第二步:请输入动物体内配方组成(配方适用于不溶于水的药物;不同批次药物配方比例不同,请联系Selleck为您提供正确的澄清溶液配方) 药物溶于 μL DMSO溶液(母液浓度 mg/mL,注:如该浓度超过该批次药物DMSO溶解度,请先联系Selleck); 体内配方配制方法:取 μL DMSO母液,加入 μL PEG300,混匀澄清后加入μL Tween 80,混匀澄清后加入 μL ddH2O,混匀澄清。 体内配方配制方法:取 μL DMSO母液,加入 μL Corn oil,混匀澄清。 注意:1. 首先保证母液是澄清的; 2. 一定要按照顺序依次将溶剂加入,进行下一步操作之前必须保证上一步操作得到的是澄清的溶液,可采用涡旋、超声或水浴加热等物理方法助溶。 本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为: 质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子量 (g/mol) 摩尔浓度计算公式 *在配置溶液时,请务必参考Selleck产品标签上、SDS / COA(可在Selleck的产品页面获得)批次特异的分子量使用本工具。 用本工具协助配置特定浓度的溶液,使用的计算公式为: 开始浓度 x 开始体积 = 最终浓度 x 最终体积 稀释公式 稀释公式一般简略地表示为: C1V1 = C2V2 ( 输入 输出 ) 在配置溶液时,请务必参考Selleck产品标签上、SDS / COA(可在Selleck的产品页面获得)批次特异的分子量使用本工具。. 连续稀释计算器方程NCT02876094 Terminated Drug: celecoxib Spinal Muscular Atrophy (SMA) Hugh McMillan|Families of Spinal Muscular Atrophy|Gwendolyn Strong Foundation|Children\'\'s Hospital of Eastern Ontario January 29 2019 Phase 2NCT03185871 Withdrawn Drug: Celecoxib Breast Carcinoma University of Wisconsin Madison|National Cancer Institute (NCI) September 20 2017 Phase 2NCT02413203 Completed Drug: Celecoxib|Drug: Placebo Healthy University of Pennsylvania|Eli Lilly and Company March 2015 Not ApplicableNCT03305068 Unknown status Drug: Celecoxib Reverse or Primary Total Shoulder|Rotator Cuff- Full Thickness- Repair St. Louis Joint Replacement Institute February 2014 Phase 4NCT02429427 Completed Drug: Celecoxib|Other: Placebo Breast Cancer Imperial College London|Institute of Cancer Research United Kingdom December 2005 Phase 3 在订购、运输、储存和使用我们的产品的任何阶段,您遇到的任何问题,均可以通过拨打我们的热线电话400-668-6834,或者技术支持邮箱tech@selleck.cn,直接联系到我们。我们会在24小时内尽快联系您。 操作手册 问题 1:I am doing an animal experiment with mice and planning to administrate S1261 via oral gavage. what are your recommendations for diluting the compound? For oral administration, Celecoxib can be dissolved in vehicle one: 0.5% methyl cellulose and 0.025% Tween-20 , or the vehicle 2 2% DMSO/30% PEG 300/5% Tween 80/ ddH2O . Non-selective COX inhibitor of COX-1 and COX-2 with IC50 of 1.23 μM and 3.50 μM, respectively. Xanthohumol,来自啤酒花的一种异戊烯化查耳酮,抑制COX-1和COX-2活性,并表现出化学预防作用。Xanthohumol 可抑制 diacylglycerol acyltransferase 1 (DGAT1) 和 DGAT2,对应的IC50值均为40 μM。Xanthohumol 也是一种有效的针对一系列DNA和RNA病毒的抗病毒药剂。Xanthohumol 在肿瘤细胞中可诱导生长阻滞和凋亡。Phase 1。 AZD3839是一种有效的选择性BACE1抑制剂,Ki为26.1 nM,比作用于BACE2的选择性高14倍。Phase 1。 Nirogacestat (PF-03084014) New Nirogacestat (PF-03084014, PF-3084014) 是一种选择性gamma-secretase抑制剂,在无细胞试验中IC50为6.2 nM。Nirogacestat (PF-03084014, PF-3084014) 可诱导凋亡。Phase 2。 Indomethacin (NSC-77541, Indometacin)是一种非选择性的COX1和COX2的抑制剂,IC50分别为0.1 μg/mL和5 μg/mL。常用于降低发热、减缓疼痛、僵硬和肿胀。 Aspirin (NSC 27223, Acetylsalicylic acid, ASA)是水杨酸类不可逆的COX1 and COX2抑制剂,常用作止痛药来缓解轻微疼痛,作为解热药减少发热,并作为一种抗炎药物。Aspirin 可诱导自噬并激发线粒体自噬。 Ketorolac是一种非选择性的COX抑制剂,作用于人类COX-1和COX-2时, IC50分别为1.23 µM和3.50 µM。 Features:Ketorolac是非类固醇类抗炎药(NSAIDs),优先抑制COX-1。 Ibuprofen (NSC 256857, Dolgesic)是一种抗炎类抑制剂,作用于COX-1和COX-2,IC50分别为13 μM和370 μM。 Features:Ibuprofen是世界卫生组织WHO基本药物清单中的核心药物, 这些药物是基本保健体系最低需求的药物清单。 Tags: 购买Celecoxib(SC 58635) | Celecoxib(SC 58635)供应商 | 采购Celecoxib(SC 58635) | Celecoxib(SC 58635)价格 | Celecoxib(SC 58635)生产 | 订购Celecoxib(SC 58635) | Celecoxib(SC 58635)代理商

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